Cholinergic Receptor

Enhancement of pharmacokinetic properties and in vivo efficacy of benzylidene ketal M2 muscarinic receptor antagonists via benzamide modification

Organic Chemistry / Pharmacokinetics / In Vitro / Humans / Animals / Drug Design / Acetylcholine / Bioavailability / Microdialysis / In Vivo / Rats / Rat / Cholinergic Receptor / Bioorganic and medicinal Chemistry / Structure activity Relationship / Muscarinic Receptor / Chemical Synthesis / Area Under Curve / Benzamides / Drug Design / Acetylcholine / Bioavailability / Microdialysis / In Vivo / Rats / Rat / Cholinergic Receptor / Bioorganic and medicinal Chemistry / Structure activity Relationship / Muscarinic Receptor / Chemical Synthesis / Area Under Curve / Benzamides

5α-cardenolides from Kanahia laniflora inhibit lonotropic acetylcholine receptors

Complementary and Alternative Medicine / Plant Biology / Pharmacognosy / Cholinergic Receptor

5α-Cardenolides from Kanahia laniflora Inhibit Ionotropic Acetylcholine Receptors

Complementary and Alternative Medicine / Plant Biology / Pharmacognosy / Patch-clamp and imaging techniques / Phytotherapy / Humans / Nicotinic Acetylcholine Receptors / Flowers / Plant extracts / Cholinergic Receptor / Apocynaceae / Plant Leaves / Humans / Nicotinic Acetylcholine Receptors / Flowers / Plant extracts / Cholinergic Receptor / Apocynaceae / Plant Leaves
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